GABA Receptor
GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. GABA receptors influence cognition by coordinating with glutamatergic processes. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels; whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors. A subclass of ionotropic GABA receptors, insensitive to typical allosteric modulators of GABAA receptor channels such as benzodiazepines and barbiturates, designated GABAС receptor.
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Phaclofen是适度的选择性 GABAB 拮抗剂。
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Pentobarbital sodium salt是Pentobarbital sodium salt enhances GABAergic activity。
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Org 20599是阳性变构的调节剂（positive allosteric modulator）且是GABAA 受体的直接激动剂。
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Ocinaplon是GABAA 调节剂，抗焦虑剂。
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NNC 711是GAT-1选择性抑制剂。
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Phaclofen是适度的选择性 GABAB 拮抗剂。
More
-
Pentobarbital sodium salt是Pentobarbital sodium salt enhances GABAergic activity。
More
-
Org 20599是阳性变构的调节剂（positive allosteric modulator）且是GABAA 受体的直接激动剂。
More
-
Ocinaplon是GABAA 调节剂，抗焦虑剂。
More
-
NNC 711是GAT-1选择性抑制剂。
More
